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Table 4 8-isopentenyl flavonoids compounds potency on PDE5A1

From: Isolation, bioassay and 3D-QSAR analysis of 8-isopentenyl flavonoids from Epimedium sagittatum maxim. as PDE5A inhibitors

Compd

PDE5A1 (IC50 ± SD) (μM)

1

8.27 ± 0.74

2

3.23 ± 0.23

3

5.47 ± 0.56

4

408.60 ± 31.4

5

357.60 ± 34.2

6

681.90 ± 38.4

Sildenafil

0.0142 ± 0.0013